| 801 |
|
Discovery and Optimization of a Novel Class of Orally Active NonpeptidicEndothelin-A Receptor Antagonists
|
Riechers, H
|
American Chemical Society
|
1980
|
|
|
|
| 802 |
|
Discovery and Preclinical Characterization of (+)-3-[4-(1-Piperidinoethoxy)phenyl]spiro[indene-1,1'-indane]-5,5'-diol Hydrochloride: A Promising Nonsteroidal Estrogen Receptor Agonist for Hot Flush/
|
Watanabe, N
|
American Chemical Society
|
2003
|
|
|
|
| 803 |
|
Discovery and Structure-Activity Relationship of Oxalylarylaminobenzoic Acids as Inhibitors of Protein Tyrosine Phosphatase 1B/
|
Liu, G
|
American Chemical Society
|
2003
|
|
|
|
| 804 |
|
Discovery and Structure-Activity Relationships of Novel Piperidine Inhibitors of Farnesyltransferase/
|
Nara, S
|
American Chemical Society
|
2003
|
|
|
|
| 805 |
|
Discovery and Synthesis of [6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]. 2-(4-hydroxyphenyl)]benzo[b]thiophene: A Novel, Highly Potent, Selective Estrogen Receptor Modulator
|
Palkowitz, A. D
|
American Chemical Society
|
1980
|
|
|
|
| 806 |
|
Discovery, Characterization, and Structure-Activity Relationships Studies of Proapoptotic Polyphenols Targeting B-Cell Lymphocyte/Leukemia-2 Proteins/
|
Kitada, S
|
American Chemical Society
|
2003
|
|
|
|
| 807 |
|
Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A)Receptor Agonist Activity. 1. Optimization of the Agonist "Trigger"
|
Aquino, C. J
|
American Chemical Society
|
1980
|
|
|
|
| 808 |
|
Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A)Receptor Agonist Activity (II): Optimization of the C3 Amino Substituent
|
Hirst, G. C
|
American Chemical Society
|
1980
|
|
|
|
| 809 |
|
Discovery of 3-Aminobenzyloxycarbonyl as an N-Terminal Group Conferring High Affinity to the Minimal Phosphopeptide Sequence Recognized by the Grb2-SH2 Domain
|
Furet, P
|
American Chemical Society
|
1980
|
|
|
|
| 810 |
|
Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido(2,3-d)-pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase Inhibitor/
|
Lee, Chih-Hung
|
American Chemical Society
|
2001
|
|
|
|
| 811 |
|
Discovery of 4-Benzoyl-1-[(4-methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)oxoace tyl]-2-(R)-methylpiperazine (BMS-378806): A Novel HIV-1 Attachment Inhibitor That Interferes with CD4-gp 120 Interactions/
|
Wang, T
|
American Chemical Society
|
2003
|
|
|
|
| 812 |
|
Discovery of Allosteric Potentiators for the Metabotropic Glutamate 2 Receptor: Synthesis and Subtype Selectivity of N-(4-(2-Methoxyphenoxy)phenyl)-N-(2,2,2-trifluoroethylsulfonyl)pyrid-3-ylmeth ylamine/
|
Johnson, M. P
|
American Chemical Society
|
2003
|
|
|
|
| 813 |
|
Discovery of an Orally Active Non-Peptide Fibrinogen Receptor Antagonist
|
Stilz, H. U
|
American Chemical Society
|
1980
|
|
|
|
| 814 |
|
Discovery of an Orally Active Series of Isoxazoline Glycoprotein IIb/IIIa Antagonists
|
Xue, C.-B
|
American Chemical Society
|
1980
|
|
|
|
| 815 |
|
Discovery of an Orally Bioavailable NK~1 Receptor Antagonist, (2S,3S)-(2-Methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with Potent Antiemetic Activity
|
Ward, P
|
American Chemical Society
|
1980
|
|
|
|
| 816 |
|
Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 1. Identification of the 4-Quinolinecarboxamide Framework
|
Giardina, G. A. M
|
American Chemical Society
|
1980
|
|
|
|
| 817 |
|
Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective �Opioid Agonists, Based on an Extension of the Message-Address Concept
|
Dondio, G
|
American Chemical Society
|
1980
|
|
|
|
| 818 |
|
Discovery of (Aryloxopropenyl)pyrrolyl Hydroxyamides as Selective Inhibitors of Class IIa Histone Deacetylase Homologue HD1-A/
|
Mai, A
|
American Chemical Society
|
2003
|
|
|
|
| 819 |
|
Discovery of a Series of Nonpeptide Small Molecules That Inhibit the Binding of Insulin-like Growth Factor (IGF) to IGF-Binding Proteins/
|
Chen, C
|
American Chemical Society
|
2001
|
|
|
|
| 820 |
|
Discovery of a Simple Picomolar Inhibitor of Cholesteryl Ester Transfer Protein/
|
Reinhard, E. J
|
American Chemical Society
|
2003
|
|
|
|